《神经系统药物 《药品集》第9分册》求取 ⇩

概述1

Ⅰ.解热镇痛药 上海医药工业研究院 沙静姝编写 蔡月刚校订1

一、水杨酸类5

1.水杨酸钠(Sodium salicylate)5

2.水杨酸钙(Calcium salicylate)5

3.水杨酰胺(Salicylamide)6

4.水杨酸甲酯(Methyl salicylate)6

5.水杨酸胆碱(Choline salicylate)7

6.三水杨酸胆三镁盐(Choline magnesium trisalicylate)7

7.乙酰水杨酸钙脲(Calicium acetylsalicylate urea)8

8.乙酰水杨酸钙(Calicium acetylsalicylate)8

9.水杨酸水杨酸酯(Salicylsalicylic acid)8

10.乙酰水杨酸(Acetyl salicylic acid)9

12.扑炎痛(Benorylate)10

一、吸入麻醉药10

11.乙酰水杨酸铝(Aluminium acetylsalicylate)10

13.乙氧基扑炎痛(Eterylate)11

14.阿司匹林赖氨酸(Aspirin-DL-lysine)11

16.氟苯水杨酸(Diflunisal)12

15.阿司匹林精氨酸(Arginine acetylsalicylate)12

17.氟苯乙酰水杨酸(Flufenisal)13

二、乙酰苯胺类13

18.乙酰苯胺(Acetanilide)13

19.醋氨酚(Acetaminophen)13

20.非那西丁(Phenacetin)14

21.乙氧苯酰胺(Ethenzamide)15

22.溴苯丙胺(Bromanyl promide)15

23.丁胺苯醚(Bucetin)16

24.苯甘胺(Ralgin)16

25.乳胺苯醚(Lactyophenetidin)17

26.桂苯氧脲(Cinnapyrin)17

28.异丙比林(Isopropylantipyrin)18

27.安替比林(Antipyrin)18

三、吡唑酮类18

29.烟酰比林(Nifenazone)19

30.胺丙比林(Aminoproylon)19

31.氨基比林(Aminopyrin)20

32.安乃近(Analgin)20

33.保泰松(Phenylbutazon)21

34.戊烯保泰松(Prenazone)22

35.羟基保泰松(Oxyphenbutazone)22

36.酮基保泰松(Ketophenylbutazone)23

37.琥珀甲酯保泰松(Suxibuzone)23

38.氯苯松(Clofezone)24

39.吖丙吡唑酮(Azapropazone)24

40.苯氧吡唑酮(Phenopyrazone)25

四、喹啉类26

41.奎宁盐酸盐(Quinine hydrochloride)26

42.奎宁梳酸盐(Quinine sulfate)26

43.碳酸乙酯奎宁(Quinine ethyl carbonate)27

44.辛可芬(Cinchophen)27

46.甲灭酸(Mefenamic acid)28

五、邻氨基苯甲酸类28

45.苯胺喹啉(Glaphenine)28

47.氟灭酸(Fulfenamic acid)29

48.氟灭酸铝盐(Aluminium flufenamate)29

49.烟氟灭酸(Niflumic acid)30

50.氯灭酸(Chlofenamic acid)30

51.甲氯灭酸(Meclofenamic acid)31

52.双氯灭酸钠(Diclofenac sodium)31

54.丙烯氯苯乙酸(Alclfenac)32

(一)烷基苯乙酸类32

六、芳基烷酸类32

53.异丁苯乙酸(Ibufenac)32

55.丁苯羟肟酸(Bufexamac)33

(二)芳基乙酸类33

56.消炎痛(Indomethacin)33

57.托耳米丁(Tolmetin)34

58.硫茚酸(Sulindac)34

59.甲嗪乙酸(Metiazinic acid)35

60.氯苯噻唑酸(Fenclozic acid)35

61.氯苯噻唑苯酸(Fentiazac)36

62.氯苯吡乙酸(Clopirac)36

63.苯甲酰吡酸钠(Zomepirac sodium dihydrate)37

(三)烷基苯丙酸类37

64.异丁苯丙酸(Ibuprofen)37

65.酮基布洛芬(Ketoprofen)38

68.苯氧布洛芬钙盐(Fenoprofen calcium)39

66.氟苯布洛芬(Flurbiprofen)39

67.吲哚布洛芬(Indoprofen)39

69.吡氯布洛芬(Pirprofen)40

70.噻吩甲酰布洛芬(Suprofen)40

72.萘普生(Naproxen)41

(四)芳基丙酸类41

71.苯乙布洛芬(Namoxyrate)41

73.苯噁布洛芬(Benoxaprofen)42

74.苯噁丙酸(Oxaprozin)42

七、其他类43

75.双苯氧酰嗪(Simetride)43

76.强痛定(Fortanodyn)43

77.氯噻哌醇(Tiaramide)44

78.甲氧嘧唑(Metopyrimazole)44

79.炎痛静(Benzydamine hydrochloride)45

80.二苯胺唑(Difenamizole)45

81.双苯甲胺乙烷(Diphenyldimethylaminoethane hydrochloride)46

82.噻嗯吡啶(Thienoridline hydrochloride)46

83.百克痛(Bucolome)47

84.苄庚唑酮(Benhepazone)48

85.湿痛喜康(Sudoxicam)48

86.炎痛喜康(Piroxicam)48

87.双酞酮(Diftalone)49

88.氯苯噁酮(Seclazone)50

89.丙喹酮(Prquazone)50

90.丁苯肼酮酸钙(Bumadizone caloium)51

91.苯酮酸(Fenbufen)51

92.氯环己茚满酸(Clidanac)51

93.三苄呋糖甙(Tribenoside)52

94.百乃定(Panadin)53

95.抗炎松(Antiflamison)53

96.铜锌过氧化物歧化酶(Orgotein)53

97.柴胡54

98.葛根54

99.淡竹叶54

八、中草药54

100.防己55

101.汉防己甲素(Tetrandrine)55

102.秦艽55

103.徐长卿56

104.威灵仙56

105.丁公藤56

109.穿山龙57

106.七叶莲57

107.卷耳子57

108.豨桐片57

110.昆明山海棠58

111.祖师麻58

112.百里香59

113.钻山风制剂59

114.安络痛59

115.健骨60

116.骨宁60

117.克痛灵60

118.蜂毒60

Ⅱ.抗痛风药 上海医药工业研究院 沙静姝编写 蔡月刚校订61

概述61

1.秋水仙碱(Colchicine)63

2.保泰松(Phenybutazone)63

一、抗痛风性关节炎急性发作药63

3.羟基保泰松(Oxyphenbutazone)64

4.消炎痛(Indomethacin)64

5.萘普生(Naproxen)64

6.苯氧布洛芬钙盐(Fenoprofen calcium)64

7.硫茚酸(Sulindac)64

(一)促进尿酸排泄剂65

9.羧苯磺胺(Probenecid)65

二、抗血中尿酸过高药物65

8.炎痛喜康(Piroxicam)65

10.苯磺唑酮(Sulfinpyrazone)66

11.酮基保泰松(Ketophenylbutazone)66

12.溴酚呋酮(Benbromarone)66

13.碘酚呋酮(Benziodarone)67

14.百克痛(Bucolome)67

15.辛可芬(Cinchophen)67

16.降脂乙酯(Clofibrate)68

17.降脂酰胺(Halofenate)68

18.醋磺环己脲(Acetohexamide)69

19.噻宁酸(Ticrynafen)69

(三)促进尿酸分解剂70

21.尿酸氧化酶70

20.别嘌醇(Allopurinol)70

(二)抑制尿酸生成剂70

Ⅲ.镇痛药 湖南医药工业研究所 上海医药工业研究院 陈国强编写 蔡月刚校订71

概述71

一、强效镇痛药72

1.吗啡(Morphine)72

2.阿片粉(Powdered opium)73

3.阿片全碱(Papaveretum)74

4.乙基吗啡(Ethylmorphine hydrochloride)74

5.苄基吗啡(Benzylmorphine hydrochloride)75

6.二乙酰吗啡(Diacetylmorphine hydrochloride)75

7.氢化吗啡酮(Hydromorphone hydrochloride)76

8.吗啡酮(Oxymorphone hydrochloride)76

9.布诺啡(Buprenorphine hydrochloride)77

10.乙烯啡(Etorphine hydrochloride)77

12.二氢可待因(Dihydrocodeine hydrogentartrate)78

11.乙酰烯啡(Acetorphine hydrochloride)78

13.二氢可待因酮(Hydrocodone hydrogentartrate)79

14.羟氢可待因酮(Oxycodone hydrochloride)79

15.左吗喃(Levorphanol tartrate)80

16.苯唑辛(Phenazocine hydrobromide)80

17.哌替啶(Meperidine hydrochloride)81

18.苯替啶(Phenoperidine hydrochloride)82

19.甲替啶(Alphaprodine hydrochloride)82

20.三甲替啶(Trimeperidine)83

21.甲哌酮(Detobemidone)83

23.安痛定(Anileridine hydrochloride)84

22.去痛定(Piminodine ethanesulfonate)84

25.哌散痛(Dipipanone hydrochloride)85

24.美散痛(Methadone hydrochloride)85

26.吗散痛(Phenadoxone hydrochloride)86

27.右吗酰胺(Dextromoramide tartrate)86

28.吗酰胺(Racemoramide)87

29.苯唑酰胺(Bezitramide)87

30.哌氰酰胺(Piritramide)88

31.芬太尼枸橼酸盐(Fentanyl citrate)88

32.二甲噻胺(Dimethylthiambutene hydrochloride)89

33.苯环己啶(Phencyclidine hydrochloride)89

34.普鲁法多(Profadol hydrochloride)90

35.甲氧异啉(Metofoline hydrochloride)90

36.太利定(Tilidine hydrochloride)91

37.镇痛利(Azabicyclane)91

38.甲氧异丁嗪(Methotrimeprazine)92

39.镇痛新(Pentazocine)92

二、弱效镇痛药93

40.可待因(Codeine phosphate)93

41.达而丰(Propoxyphene hydrochloride)94

42.乙氧庚嗪枸橼酸盐(Ethoheptazine citrate)94

43.乙氧酰胺(Carbiphene hydrochloride)95

44.苯吡胺醇(Phenyramidol hydrochloride)95

45.延胡索乙素(Tetrahydropalmatine)96

46.颅通定(Rotundine)96

48.七叶莲97

47.延胡索97

三、镇痛中草药97

49.木通七叶莲98

50.牛藤98

51.野木瓜98

52.鸡屎藤98

53.华千金藤99

54.徐长卿99

55.白屈菜99

56.雪上一枝蒿100

57.毛蒟100

58.安络痛100

1.丙烯吗啡(Nalorphine hydrochloride)101

概述101

〔附〕吗啡受体拮抗剂101

59.祖师麻101

2.丙烯左吗南(Levallorphan tartrate)102

3.丙烯吗啡酮(Naloxone hydrochloride)103

4.环唑辛(Cyclazocine)103

5.环丙烯啡(Cyprenorphine)104

Ⅳ.全身麻醉药 广东医药工业研究所 上海医药工业研究院 霍景文 蔡月刚 编写 蔡月刚校订105

概述105

1.氧化亚氮(Nitrous oxide)107

2.乙醚(Ether)107

3.乙烯醚(Vinyl ether)108

4.乙基乙烯醚(Ethyl vinyl ether)108

6.乙烯(Ethylene)109

5.环丙烷(Cyclopropane)109

7.三氯乙烯(Trichloroethylene)110

8.氟烷(Halothane)110

9.甲氧氟烷(Methoxyflurane)111

10.三氟乙基乙烯醚(Fluroxene)111

11.安氟醚(Enflurane)112

12.异氟醚(Isoflurane)112

13.氯仿(Chloroform)113

14.氯乙烷(Ethyl chloride)113

二、静脉麻醉药114

15.硫喷妥钠(Thiopental sodium)114

16.丙烯硫喷妥钠(Htiamylal sodium)114

18.甲基环己烯巴比妥钠(Hexobarbital sodium)115

17.硫代烯丙巴比妥钠(Thiabarbital sodium)115

19.丙烯炔巴比妥钠(Methohexital sodium)116

20.安定(Diazepam)116

21.氟硝安定(Flunitrazepam)117

22.羟丁酸钠(Sodium oxybate)118

23.普尔安(Propanidid)118

24.氯胺酮(Ketamine hydrochloride)119

25.羟孕酮琥珀酸酯钠(Hydroxydione sodium succinate)120

26.爱舒新(Althesin)120

27.乙咪酯(Etomidate sulfate)121

28.氟哌啶(Droperidol)122

29.芬太尼枸橼酸盐(Fentanyl citrate)122

31.副醛(Paraldehyde)123

30.三溴乙醇(Tribromoethanol)123

三、直肠麻醉药123

Ⅴ.局部麻醉药 广东医药工业研究所 郑宽 霍景文 编写 郑宽校订124

概述124

一、酯类125

1.普鲁卡因(Procaine hydrochloride)125

2.氯普鲁卡因(Chloroprocaine hydrochloride)126

3.丁氧普鲁卡因(Benoxinate hydrochloride)126

4.可卡因(Cocaine hydrochloride)127

5.丁卡因(Tetracaine hydrochloride)128

6.戊氨卡因(Naepaine hydrochloride)129

7.丁氨卡因(Butethamine hydrochloride)129

9.丙氧卡因(Propoxycaine hydrochloride)130

8.布大卡因(Butacaine sulfate)130

10.苯佐卡因(Benzocaine)131

11.氨苯丁酯(Butyl aminobenzoate)131

12.氨苯异丁酯(Isobutyl aminobenzoate)132

13.亮卡因甲磺酸盐(Leucinoeaine mesylate)132

14.杜土卡因(Tutoeaine hydrochloride)132

15.间丁乙胺(Metabutethamine hydrochloride)133

16.间丁氧卡因(Metabutoxyeaine hydrochloride)133

17.丙对卡因(Proparacaine hydrochloride)134

18.凹索卡因(Orthocaine)134

19.异戊卡因(Amylocaine hydrochloride)135

20.哔哌卡因(Piperocaine hydrochloride)135

22.己卡因(Hexylcaine hydrochloride)136

21.环甲卡因(Cyclomethycaine sulfate)136

23.异丁卡因(Isobucaine hydrochloride)137

24.阿米德里卡因(Amydricaine hydrochloride)137

25.托派古柯碱(Tropacocaine hydrochloride)138

26.苯扎明(Benzamine hydrochloride)138

27.甲丙卡因(Meprylcaine hydrochloride)139

二、酰胺类139

28.利多卡因(Lidocaine hydrochloride)139

29.丙胺卡因(Prilocaine hydrochloride)140

30.地布卡因(Dibucaine hydrochloride)141

31.衣铁卡因(Etidocaine hydrochloride)142

32.丁哌卡因(Bupivacaine hydrochloride)142

33.吡甲卡因(Pyromocaine hydrochloride)143

34.甲哌酰卡因(Mepivacaine hydrochloride)144

35.阿泊土卡因(Aptocaine hydrochloride)145

36.甲苯卡因(Tolycaine hydrochloride)145

37.羟乙卡因(Oxethacaine)145

38.吡咯卡因(Pyrrocaine hydrochloride)146

39.三甲卡因(Trimecaine hydrochloride)147

40.庚卡因(Heptacaine hydrochloride)147

41.丁苯胺卡因(Butanilicaine hydrochloride)148

42.甲基丙胺卡因(Quatacaine hydrochloride)148

43.狄帕洛东(Diperodon hydrochloride)149

三、其他类型149

44.达克罗宁(Dyclonine hydrochloride)149

45.丙吗卡因(Pramoxine hydrochloride)150

46.丁吖啶(Centbucridine hydrochloride)150

47.酮卡因(Ketocaine)151

48.异喹卡因(Dimethisoquin hydrochloride)152

49.非那卡因(Phenacaine hydrochloride)152

50.苯甲醇(Benzyl alcohol)153

51.水杨醇(Salicyl alcohol)153

52.丁香酚(Eugenol)153

53.胺苯呋酮(Amolanone hydrochloride)154

54.己硫卡因(Hexothiocaine hydrochloride)154

55.优库平(Euprocin hydrochloride)155

56.局麻宁155

Ⅵ.镇静催眠药 湖南医药工业研究所 上海医药工业研究院 上海医药工业研究院 陈国强 蔡月刚 编写 蔡月刚校订156

概述156

1.巴比妥(Barbital)160

一、巴比妥类160

2.巴比妥钠(Barbital sodium)161

3.苯巴比妥(Phenobarbital)161

4.苯巴比妥钠(Phenobarbital sodium)162

5.甲基巴比妥(Metharbital)162

6.甲基苯巴比妥(Mephobarbital)163

7.苯甲巴比妥(Heptobarbital)163

8.二烯丙比巴比妥(Allobarbital)164

9.异戊巴比妥(Amobarbital)164

10.异戊巴比妥钠(Amobarbital sodium)165

11.戊巴比妥钠(Pentobarbital sodium)165

12.戊巴比妥钙(Pentobarbital calcium)166

13.丁巴比妥(Butobarbital)166

15.戊烯巴比妥钠(Vinbarbital sodium)167

14.另丁巴比妥钠(Butabarbital sodium)167

17.烯异丙巴比妥(Aprobarbital)168

16.戊烯巴比妥(Vinbarbital)168

18.溴烯异丙巴比妥(Propallylonal)169

19.烯丁巴比妥(Talbutal)169

20.烯异丁巴比妥(Butalbital)169

21.烯新戊巴比妥(Nealbarbital)170

22.环己烯巴比妥钙(Cyclobarbital calcium)170

23.环己烯巴比妥(Cyclobarbital)171

24.甲基环己烯巴比妥(Hexobarbital)171

25.烯戊巴比妥钠(Secobarbital sodium)172

26.烯戊巴比妥(Secobarbital)172

28.氟安定(Flurazepam hydrochloride)173

27.环庚烯巴比妥(Heptabarbital)173

三、苯并二氮杂？类173

29.硝基安定(Nitrazepam)174

30.舒乐安定(Estazolam)174

31.三唑安定(Triazolam)175

三、其他类176

32.乌拉坦(Urethan)176

33.炔己蚁胺(Ethinamate)176

34.丙炔蚁胺(Hexapropymate)177

35.水合氯醛(Cholral hydrate)177

36.丁基氯醛(Butylchloral hydrate)178

37.氯醛甜碱(Chloral betaine)178

39.氯醛酰胺(Chloralformamide)179

38.氯醛比林(Dichloralphenazon)179

40.氯醛葡糖(Chloralose)180

41.羟环氯醛(Penthrichloral)180

42.三氯磷酯钠(Triclofos sodium)180

43.氯丁醇(Chlorobutanol)181

44.氯己醇(Chlorhexadol)181

45.副醛(Paraldehyde)182

46.叔戊醇(Amylene hydrate)182

47.乙氯炔醇(Ethchlorvynol)183

48.甲戊炔醇(Methylpentynol)183

50.甲乙眠砜(Methylsulfonal)184

51.乙溴酰脲(Carbromal)184

49.二乙眠砜(Sulfonal)184

52.乙酰溴脲(Acetylcarbromal)185

53.溴戊酰脲(Bromisovalum)185

54.乙丁酰脲(Eetylurea)186

55.丙戊酰脲(Apronal)186

56.氨甲丙二酯(Meprobamate)186

57.苯乙哌酮(Glutethimide)187

58.甲乙哌酮(Methyprylon)188

59.安眠酮(Methaqualone)188

60.甲哌淀(Perlapine)189

61.氯甲噻唑乙烷二磺酸盐(Chlormethiazole edisylate)189

62.溴化钠(Sodium bromide)190

63.溴化钾(Potassium bromide)190

66.一溴樟脑(Bromcamphora)191

65.溴化钙(Calcium bromide)191

64.溴化铵(Ammonium bromide)191

67.缬草酸(Valeric acid)192

68.缬草192

69.朱砂192

70.远志193

71.酸枣仁193

72.合欢皮193

73.柏子仁194

74.瓜子金194

75.石菖蒲194

76.首乌195

77.丹参195

78.黄花败酱196

Ⅷ.抗精神病药 湖南医药工业研究所 上海医药工业研究院 陈国强 蔡月刚 编写 蔡月刚校订197

概述197

一、吩噻嗪类199

1.氯丙嗪(Chlorpromzine hydrochloride)199

2.乙氯丙嗪(Chlorproethazine)200

3.哌氯丙嗪(Pipamazine)200

4.氯丙嗪亚砜(Chlorpromazine sulfoxide)201

5.丙嗪(Promazine hydrochloride)201

6.乙酰丙嗪(Acepromazine maleate)202

7.三氟丙嗪(Triflupromazine hydrochloride)202

8.异丁嗪(Trimeprazine tartrate)203

9.甲氧异丁嗪(Methotrimeprazine)203

11.氨砜拉嗪(Thioproperazine dimethanesulfonate)204

10.三氟拉嗪(Trifluoperazine dihydrochloride)204

12.丙拉嗪(Perazine)205

13.氯拉嗪(Prochlorperazine dimaleate)205

14.丁酰拉嗪(Butaperazine maleate)206

15.乙硫拉嗪(Thiethylperazine dimaleate)206

16.丁羟拉嗪(Dixyrazine dihydrochloride)207

17.奋乃静(Perphenazine)208

18.乙酰奋乃静(Acetophenazine dimaleate)208

19.丙酰奋乃静(Carphenazine dimaleate)209

20.三甲氧奋乃静(Methophenazine)209

21.奋乃静乙酯(Thiopropazate dihydrochloride)210

22.氟奋乃静(Fluphenazine dihydrochloride)210

24.氟奋乃静癸酸酯(Fluphenazine decanoate)211

23.氟奋乃静庚酸酯(Fluphenazine enanthate)211

25.氧氟奋乃静(Oxaflumazine disuccinate)212

26.甲硫哒嗪(Thioridazine hydrochloride)212

27.甲砜哒嗪(Mesoridazine besylate)213

28.密哌嗪(Mepazine hydrochloride)213

29.哌乙酰嗪(Piperacetazine)214

30.氰噻嗪(Pericyazine)215

31.哌甲氧嗪(Perimetazine)215

32.哌普嗪十一烯酸酯(Pipotiazine undecylenate)215

33.哌普嗪棕榈酸酯(Pipotiazine palmitate)216

34.螺环氯嗪(Spiclomazine hydrochloride)216

35.吡啶丙嗪(Prothipendyl hydrochloride)217

37.氯噻吨(Clopenthixol)218

二、硫杂蒽类218

36.泰尔登(Chlorprothxene)218

38.氨砜噻吨(Thiothixene)219

39.三氟噻吨(Flupenthixol dihydrochloride)219

40.三氟噻吨癸酸酯(Flupenthixol decanoate)220

三、丁酰苯类220

41.氟哌丁苯(Haloperidol)220

42.三氟哌丁苯(Trifluperidol)221

43.氯氟哌丁苯(Clofluperol)221

44.甲哌丁苯(Moperone hydrochloride)222

45.酰胺哌丁苯(Pipamperone dihydrochloride)222

47.螺环哌丁苯(Spiperone)223

46.甲氧哌丁苯(Fluanisone)223

48.氟哌啶(Droperidol)224

49.咪哌丁苯(Benperidol)224

50.丙氨哌丁苯(Carperone)225

四、利血平类225

51.利血平(Reserpine)225

52.去甲氧利血平(Deserpidine)226

53.桂皮利血胺(Pescinnamine)226

五、其他227

54.碳酸锂(Lithium carbonate)227

55.氟乙醚(Flurothyl)228

56.氯噻平(Clothiapine)228

57.氯氮平(Clozapine)228

59.甲硫平(Metiapine)229

58.甲氯氧平琥珀酸盐(Loxapine succinate)229

60.氯丙啶(Clomacran)230

61.舒必利(Sulpiride)230

62.吲哌啶(Oxypertine)231

63.氮甲环醇(Azacyclonol hydrochloride)231

64.三甲氯啉(Trimetozine)232

65.丁苯嗪(Tetrabenazine)232

66.卡哌咪嗪(Carpipramine)233

67.氯哌咪嗪(Clocapramine dihydrochloride)233

68.哌迷清(Pimozide)234

69.五氟利多(Penfluridol)234

70.氟斯必灵(Fluspirilene)235

71.吗啉酮(Molindone)235

73.洋金花236

72.马桑寄生236

74.黄芫花237

75.京大戟237

Ⅷ.抗忧郁药物 湖南医药工业研究所 上海医药工业研究院 陈国强 蔡月刚 编写 蔡月刚校订239

概述239

一、三环抗忧郁药240

1.丙咪嗪(Imipramine hydrochloride)240

2.丙咪嗪氧(Imipramine N-oxidehydrochloride)241

3.去甲丙咪嗪(Desipramine hydrochloride)241

4.甲丙咪嗪(Trimipramine maleate)242

5.氯丙咪嗪(Clomipramine hydrochloride)243

6.丙咪嗪酮(Ketipramine fumarate)243

8.去甲替林(Nortriptyline hydrochloride)244

7.阿密替林(Amitriptyline hydrochloride)244

9.普罗替林(Protriptyline hydrochloride)245

10.氮氧替林(Noxiptiline hydrochloride)245

11.多虑平(Doxepin hydrochloride)246

12.多硫平(Dothiepin hydrochloride)246

13.阿丙哌醇(Opipramol dihydrochloride)246

14.二甲丙蒽(Melitracen hydrochloride)247

15.甲丙吖啶(Dimethacrin tartrate)247

16.二苯氮平(Dibenzepin hydrochloride)248

17.氯氧平(Amoxapine)248

18.胺丙哚(Iprindole hydrochloride)249

二、四环和双环抗忧郁药249

19.麦普替林(Maprotiline hydrochloride)249

20.甲庚吡嗪(Mianserin hydrochloride)250

21.苯氧吗啉(Viloxazine hydrochloride)251

22.溴苯丙啶(Zimelidine)251

三、单胺氧化酶抑制剂252

23.异噁酰肼(Isocarboxaxid)252

24.尼亚酰胺(Nialamide)252

25.苯乙肼(Phenelzine)253

26.胡椒异丙肼(Safrazine)253

27.苯异丙肼(Pheniprazine hydrochloride)254

28.异丙烟肼(Iproniazid phosphate)254

29.甲苄肼(Mebanazine)255

30.苯氧丙肼(Phenozypropazine hydrogen maleate)255

31.苯环丙胺(Tranylcypromine sulfate)255

32.苯丙胺(Amphetamine sulfate)256

四、苯丙胺类和其他精神运动兴奋剂256

33.右旋苯丙胺(Dextroamphetamine sulfate)257

34.甲基苯丙胺(Methamphetamine hydrochloride)257

35.哌甲酯(Methylphenidate hydrochloride)258

36.匹莫林(Pemoline)258

37.哌苯甲醇(Pipradrol hydrochloride)259

38.氨苯异喹(Nomifensine)260

39.苯戊吡烷(Prolintane hydrochloride)260

40.氯酯醒(Meclofenoxate hydrochloride)261

41.甲苄氧胺(Tofenacin hydrochloride)261

43.氯苯戊醇(Fenpentadiol)262

44.三唑酮(Trazodone hydrochloride)262

42.L-5-羟色氨酸(L-Hydroxytryptophan)262

Ⅸ.抗焦虑药物 湖南医药工业研究所 上海医药工业研究院 陈国强编写 蔡月刚校订264

概述264

一、苯并二氮杂？类265

1.利眠宁(Chlordiazepoxide hydrochloride)265

2.安定(Diazepam)266

3.去甲羟基安定(Oxazepam)266

4.羟基安定(Temazepam)267

5.去氧安定(Medazepam)267

6.氯羟安定(Lorazepam)268

7.溴安定(Bromazepam)268

8.氟乙安定(Halazepam)269

9.三氟安定(Triflubazam)269

11.噁嗪安定(Ketazolam)270

10.噁唑安定(Oxazolam)270

12.氯唑安定(Cloxazolam)271

13.环丙安定(Prazepam)271

14.安定羟酸钾盐(Clorazepate dipotassium)272

15.氯噻安定(Clotiazepam)272

二、丙二醇类273

16.氨甲丙二酯(Meprobamate)273

17.氨甲丁二酯(Mebutamate)273

18.丁氨丙二酯(Tybamate)274

19.氨甲己酯(Emylcamate)274

20.环戊氨酯(Cyelarbamate)275

三、二苯甲烷类275

21.羟嗪(Hydroxyzine hydrochloride)275

23.丁硫乙胺(Captodiamine hydrochloride)276

22.氯苯丁嗪(Buclizine hydrochloride)276

24.苯羟乙胺(Benactyzine hydrochloride)277

25.苯羟哌啶(Pipethanate hydrochloride)277

四、其他类278

26.氯甲噻酮(Chlormezanone)278

27.羟苯丁酯(Hydroxyphenamate)278

28.苯丙氨酯(Phenprobamate)279

29.氯苯丁醇(Phenaglycodol)279

30.甲氧噁酮(Mephenoxalone)279

31.环氧酰胺(Oxanamide)280

32.戊甲酰胺(Valnoctamide)280

33.苯嗪酰胺(Benzquinamide)281

34.苯辛胺(Benzoctamine hydrochloride)281

概述282

Ⅹ.抗震颤麻痹药 上海医药工业研究院 蔡月刚、殷瑞华编写 蔡月刚校订282

一、增加脑内多巴胺药283

1.左旋多巴(Levodopa)283

2.甲多巴肼(Carbidopa)284

3.苄丝肼(Benserazide hydrochloride)285

4.金刚烷胺(Amantadine hydrochloride)285

5.左旋苯炔胺(L-deprenyl)286

二、抗胆碱药286

6.苯海索(Benzhexol hydrochloride)286

7.卡马特灵(Procyclidine hydrochloride)287

8.环戊哌醇(Cycrimine hydrochloride)288

9.双环庚啶(Biperiden hydrochloride)288

11.乙苄托品(Ethybenztropine hydrochloride)289

10.苄托品甲磺酸盐(Benztropine mesylate)289

12.东茛菪碱氢溴酸盐(Hyoscine hydrochloride)290

13.乙胺丙嗪(Ethopropazine hydrochloride)291

14.苯海拉明(Diphenhydramine hydrochloride)291

16.氯苯氧胺(Chlorphenoxamine hydrochloride)293

17.苯醇酸胺(Benapryzine hydrochloride)293

18.胺丙吗啶双环己氨基磺酸盐(Elantrine dicyclohexylsulfamate)294

三、其他治疗药294

19.溴麦角隐碱甲磺酸盐(Bromocriptine mlesylate)294

20.多巴哌酮(Domperidone hydrochloride)295

Ⅺ.抗癫痫药 上海医药工业研究院 蔡月刚、殷瑞华编写 蔡月刚校订296

概述296

1.苯妥英钠(Phenytoin sodium)298

一、乙内酰脲类298

2.甲妥因(Mephenytoin)299

3.乙妥因(Ethotoin)300

4.苯乙妥因(Phenylethylhydantoin)300

5.丁硫妥因(Albutoin)301

二、巴比妥类301

6.苯巴比妥(Phenobarbital)301

7.去氧苯巴比妥(Primidone)302

8.甲基苯巴比妥(Mephobarbital)302

9.甲基巴比妥(Metharbital)303

10.异戊巴比妥(Amobarbital)303

11.氨苯谷酰胺(Aminoglutethimide)303

三、噁唑烷酮类304

12.三甲双酮(Trimethadione)304

14.二甲双酮(Dimethadione)305

四、琥珀酰胺类305

15.乙琥胺(Ethosuximide)305

13.对甲双酮(Paramethadione)305

16.甲琥胺(Methsuximide)306

17.苯琥胺(Phensuximide)306

五、乙酰脲类307

18.苯乙酰脲(Phenacemide)307

20.乙酰苯丁酰脲(Acetylpheneturide)308

21.苄氯丙酰胺(Beclamide)308

19.苯乙酰脲(Pheneturide)308

22.安定(Diazepam)309

23.硝基安定(Nitrazepam)309

六、苯并二氮杂？类309

24.氯硝安定(Clonazepam)310

七、其他药物310

25.丙戊酸钠(Valproate sodium)310

26.卡巴咪嗪(Carbamazepine)311

27.醋氮酰胺(Acetazolamide)311

28.甲醋唑胺(Methazolamide)312

29.硫噻嗪(Sulthiame)312

30.水合氯醛(Chloral hydrate)313

31.副醛(Paraldehyde)313

32.氨甲丙二酯(Meprobamate)314

33.抗癫灵(Antiepilepsirine)314

34.阿的平(Atebrin hydrochloride)314

37.钩藤315

35.全蝎315

36.蜈蚣315

38.天麻316

Ⅻ.中枢兴奋药 上海医药工业研究院 沙静姝编写 蔡月刚校订317

概述317

1.咖啡因(Caffeine)318

2.咖啡因苯甲酸钠(Caffeine sodium benzoate)318

一、大脑兴奋药318

4.咖啡因枸橼酸盐(Caffeine citrate)319

5.羟丙茶碱(Dyphylline)319

3.甲基咖啡因(Methylcaffeine)319

7.尼可刹平(Nikethamide)320

6.印防己毒素(Picrotoxin)320

8.戊四氮(Pentylenetetrazol)320

二、延髓兴奋药320

9.回苏灵(Dimefline)321

10.贝美格(Bemegride)321

11.益迷奋(Ethamivan)322

12.双吗啉胺(Dimorpholamine)322

13.吗乙本咯(Doxapram hydrochloride)323

14.氟乙醚(Flruothyl)323

15.樟脑(Camphor)324

16.氧化樟脑(Vitacampher)325

17.来西蟾酥毒素(Resibufogenin)325

18.东茛菪碱(Scopolamine)326

19.二氧化碳(Carbon dioxide)326

三、脊髓兴奋药327

21.细胞色素丙(Cytochrome C)327

22.士的宁(Strychnine nitrate)327

20.氧(Oxygen)327

23.一叶萩碱(Securinine)328

24.野靛碱(Cytisine)329

25.山梗菜碱(Lobeline)329

四、反射性兴奋药329

五、其他330

27.氨氢吖啶(Tacrine)330

26.氨(Ammonia)330

30.人参331

六、中草药331

31.刺参酊331

29.匹莫林(Pemoline)331

28.哌甲酯(Methylphenidate hydrochloride)331

34.鹿草根332

33.柯拉子332

35.醒脑静332

32.五味子332

概述333

1.脑复新(Pyrithioxin hydrochloride)333

XIII.脑代谢功能活化剂 上海医药工业研究院 沙静姝编写 蔡月刚校订333

2.氨酪酸(γ-Aminobutyric acid)334

3.羟基氨酪酸(γ-Amino-β-hydroxybutyric acid)334

5.克脑迷(Antiradon)335

6.胞二磷胆碱(Citicoline)335

4.氯酯醒(Mcclofenoxate hydrocholride)335

7.脑复康(Piracetam)336

8.己酮可可碱(Pentoxifylline)337

9.肉桂苯哌嗪(Cinnarizine)337

10.环扁桃酯(Cyclandelate)338

11.氢化麦角毒碱甲烷磺酸盐(Dihydroergotoxine mesylate)338

12.乙酰谷酰胺(Aceglutamide)339

13.烟胺乙酯(Nicametate)339

XIV.骨骼肌、平滑肌松驰药 广东医药工业研究所 郑宽 霍景文 编写 郑宽校订341

概述341

(一)非去极化型345

1.氯化筒箭毒碱(Tubocurarine chloride)345

一、骨骼肌松驰药345

2.氟化二甲筒箭毒碱(Mecostrin chloride)346

3.碘化二甲筒箭毒碱(Metocurineiodide)346

4.三碘季铵酚(Gallamine triethiodide)347

5.潘寇罗宁(Pancuronium bromide)348

6.达冠罗宁(Dacuronium bromide)349

7.诺寇隆(Norcuron)350

8.安特寇林(Atracurium besylate)350

9.氯化亚松安(Alcuronium chloride)351

10.双苯偶氮咪唑(Fazadinium bromide)352

11.双甲偶氮咪唑(AH 10407)352

12.肌安松(Paramyon)353

13.劳多利新(Laudexium methylsulphate)354

14.瓢箭毒碱(C-Toxiferine Ⅰ)354

(二)去极化型355

16.氯化琥珀胆碱(Suxamethonium chloride)355

15.双巴辛(Diplacine hydrochloride)355

17.溴化琥珀胆碱(Suxamethonium bromide)357

19.溴化琥珀乙基胆碱(Suxamethonium bromide)358

20.溴化十烃双铵(Decamethonium bromide)358

18.碘化琥珀胆碱(Suxamethonium iodide)358

21.碘化十烃双铵(Decamethonium iodide)359

(三)双相型360

23.己氨胆碱(Carbolonium bromide)360

22.溴化六芴(Hexafluorenium bromide)360

(四)混合型361

25.醌肌松(Benzoquinonium chloride)361

24.泼瑞司通(Prodeconium bromide)361

(五)中草药362

26.汉肌松(Metetrandrine iodide)362

27.溴甲素(Metetrandrine bromide)363

28.汉松敏(Fangchinoline dimethobromide)364

29.汉己素(Cyclanoline)365

30.傣肌松(Hayatin methiodide)365

31.银不换366

32.海轮碱Ⅱ(ο,ο-Dimethyl-τ-curine dimethyl cchloride)367

33.ι-筒箭毒碱磺甲烷盐(ι-Curine methyl iodide)368

34.粉背轮环藤369

35.环轮宁双碘甲烷盐(Cycleanine dimethyl iodide)369

36.华千金藤370

37.黔桂千金藤370

39.长根金不换371

40.八角枫碱(Aunbasine hydrochloride)371

38.山豆根371

41.瓜木372

43.野花椒根373

44.蛇足草373

42.山花椒373

45.大花飞燕草374

46.绢毛高翠雀花碱(Elatine)374

48.野黑豆375

49.溴化甲基延胡索乙素(Rotundin methyl bromide)375

47.蘗肌松(Meberbamine iodide)375

50.厚朴376

51.头花千金藤376

二、作用于中枢的肌肉松驰药(包括平滑肌松驰药)377

52.美乃星(Mephenesin)377

53.美乃星氨基甲酸酯(Mephenesin carbamate)378

54.舒筋灵(Methocarbamol)378

55.氯乃星氨基甲酸酯(Chlorphenesin carbamate)379

56.利眠宁(Chlordiazepoxide hydrochloride)379

57.安定(Diazepam)380

58.环丙安定(Prazepam)381

60.安适定(Alprazolam)382

61.氯甲噻酮(Chlormezanone)382

59.松肌定(Tetrazepam)382

62.甲氧噁酮(Mephenoxalone)383

63.二苯胺唑(Difenamizole)383

64.氨甲丙二酯(Meprobamate)384

65.卡来锑(Carisoprodol)384

66.氨甲己酯(Emylcamate)385

67.氯噁唑(Chlorzoxazone)385

68.痉痛停(Tizanidine)386

69.间沙龙(Metaxalone)386

70.舒拉美(Styramate)387

71.邻甲拉明枸橼酸盐(Orphenadrine citrate)387

72.邻甲拉明(Orphenadrine hydrochloride)388

73.肌舒平(Nefopam hydrochloride)388

74.美肌松(Tolperisone hydrochloride)389

75.苯丙氨酯(Phenprobamate)390

76.苯哌醇甲磺酸盐(Pridinol methanesulfonate)390

77.苯咪唑(Benzimidzole)391

78.环戊氨酯(Cyclarbamate)392

79.疼脱龙(Dantrolene sodium)392

80.拜克罗芬(Baclofen)393

81.氯苯氧胺(Chlorphenoxamine hydrochloride)394

82.环苯庚烯(Cyclobenzaprine hydrochloride)394

83.苯辛胺(Benzoctamine hydrochloride)395

84.羟乙肉桂酰胺(Idrocilamide)395

86.哌氧酮(Pipoxolan hydrochloride)396

87.葡硫秋水仙碱(Thiocolchicoside)396

85.苯吡胺醇(Phenyramidol hydrochloride)396

88.缓肌嗪(Meladrazine)397

89.茶碱(Theophylline)397

90.氨茶碱(Aminophylline)399

91.胆茶碱(Choline theophyllinate)400

92.羟丙茶碱(Dyphylline)400

93.氨异丁醇茶碱(Ambuphylline)401

94.二乙氨乙茶碱(Etamiphyllin camsylate)401

95.罂粟碱(Papaverine hydrochloride)402

96.卡马特灵(Procyclidine hydrochloride)402

97.羟苄麻黄碱(Ritodrine hydrochloride)403

98.黄酮哌酯(Flavoxate hydrochloride)403

99.胺丙噁二唑枸橼酸盐(Proxazole oitrate)404

100.麦皮凡林(Mebeverine hydrochloride)404

101.痛灭舒达(Tolmesoxide)405

概述406

1.加兰他敏(Galanthamine hydrobromide)406

XV.骨骼肌、平滑肌兴奋药 广东医药工业研究所 上海医药工业研究所 霍景文 沙静姝编写 沙静姝校订406

2.溴化新斯的明(Neostigmine bromide)407

3.新斯的明甲基硫酸盐(Neostigmine methylsulfate)408

4.溴化嗓啶斯的明(Pyridostigmine bromide)408

5.双斯的明(Distigmine bromide)409

6.酶抑宁(Ambenonium chloride)409

7.氯化腾喜龙(Edrophonium chloride)410

9.溴化苄基吡啉(Benzpyrinium bromide)411

10.氯化乙酰胆碱(Acetylcholine chloride)411

8.氨氢吖啶(Tacrine)411

11.氯化乙酰甲胆碱(Methacholine chloride)412

12.溴化乙酰甲胆碱(Methacholine bromide)413

13.氯化氨甲酰胆碱(Carbachol)413

14.氯化氨甲酰甲胆碱(Bethanechol chloride)414

15.氯化乙酰丙胆碱(γ-Butyrobetaine chloride methyl ester)414

16.酰喹核水杨酸盐(Aceclidine salicylate)415

17.双异丙氟磷酸酯(Isofluorphate)415

18.乙硫磷(Echothiophate iodide)416

19.四乙基焦磷酸酯(Tetraethyl pyrophosphate)416

20.辛甲焦磷酰胺(Octamethyl pyrophosphoramide)417

主要参考文献418

中文索引419

外文索引430

15.邻甲拉明(Orphenadrine hydrochloride)922